Author: Karl A. Scheidt
Publisher:
ISBN:
Category :
Languages : en
Pages : 652
Book Description
I. Design and Synthesis of Cysteine Protease Inhibitors. II. Total Synthesis of (-)-bafilomycin A1 III. Studies Directed Towards the Total Synthesis of Apoptolidin
Author: Karl A. Scheidt
Publisher:
ISBN:
Category :
Languages : en
Pages : 652
Book Description
Publisher:
ISBN:
Category :
Languages : en
Pages : 652
Book Description
Studies on the Total Synthesis of Tetrafibricin ; Synthesis of Conformationally Constrained Cysteine Protease Inhibitors ; Palladium Catalyzed Synthesis of N-aryl-2-benzylindolines Via Tandem Arylation of 2-allylaniline(s)
Author: Ricardo Lira
Publisher: ProQuest
ISBN: 9780549723523
Category : Cysteine proteinases
Languages : en
Pages : 466
Book Description
Detailed in the following thesis are: (1) the diastereoselective synthesis of the C(1)-C(19) fragment of tetrafibricin, (2) a convenient, direct method for the synthesis 1,5-syn-(E)-diols from aldehyde precursors, and (3) application of this method to the completion of the C(23)-C(40) fragment of tetrafibricin (this transformation involves an initial allylboration generating syn-[beta]-alkoxyallylstannane intermediates, followed by an allylstannation step), (4) The synthesis of the complete C(1)-C(40) fragment via our double allylboration strategy and efforts towards the total synthesis of tetrafibricin, (5) the development of a convenient method to access syn-[beta]-hydroxyallylsilanes via a Lewis acid-promoted [gamma]-silylallylboration of alipathic aldehydes with new (Z)-[gamma]-silylallylboronate reagents, (6) The synthesis of a new class of conformationally constrained cysteine protease inhibitors via ring closing metathesis step, (7) a palladium-catalyzed synthesis of N-aryl-2-benzylindolines via a tandem arylation of 2-allylanilines, (this transformation leads to the formation of two C-N bonds and one C-C bond in a one-pot process, and high selectivity is observed for the sequential installation of two different aryl groups).
Publisher: ProQuest
ISBN: 9780549723523
Category : Cysteine proteinases
Languages : en
Pages : 466
Book Description
Detailed in the following thesis are: (1) the diastereoselective synthesis of the C(1)-C(19) fragment of tetrafibricin, (2) a convenient, direct method for the synthesis 1,5-syn-(E)-diols from aldehyde precursors, and (3) application of this method to the completion of the C(23)-C(40) fragment of tetrafibricin (this transformation involves an initial allylboration generating syn-[beta]-alkoxyallylstannane intermediates, followed by an allylstannation step), (4) The synthesis of the complete C(1)-C(40) fragment via our double allylboration strategy and efforts towards the total synthesis of tetrafibricin, (5) the development of a convenient method to access syn-[beta]-hydroxyallylsilanes via a Lewis acid-promoted [gamma]-silylallylboration of alipathic aldehydes with new (Z)-[gamma]-silylallylboronate reagents, (6) The synthesis of a new class of conformationally constrained cysteine protease inhibitors via ring closing metathesis step, (7) a palladium-catalyzed synthesis of N-aryl-2-benzylindolines via a tandem arylation of 2-allylanilines, (this transformation leads to the formation of two C-N bonds and one C-C bond in a one-pot process, and high selectivity is observed for the sequential installation of two different aryl groups).
American Doctoral Dissertations
Author:
Publisher:
ISBN:
Category : Dissertation abstracts
Languages : en
Pages : 848
Book Description
Publisher:
ISBN:
Category : Dissertation abstracts
Languages : en
Pages : 848
Book Description
Selected Studies in Asymmetric Synthesis
Author: William John Smith (III.)
Publisher:
ISBN:
Category :
Languages : en
Pages : 542
Book Description
Publisher:
ISBN:
Category :
Languages : en
Pages : 542
Book Description
Studies Towards the Total Synthesis of Bafilomycin A1
Author: Iain Simpson
Publisher:
ISBN:
Category :
Languages : en
Pages :
Book Description
Publisher:
ISBN:
Category :
Languages : en
Pages :
Book Description
Dissertation Abstracts International
Author:
Publisher:
ISBN:
Category : Dissertations, Academic
Languages : en
Pages : 992
Book Description
Publisher:
ISBN:
Category : Dissertations, Academic
Languages : en
Pages : 992
Book Description
I. Studies Toward the Total Synthesis of Scytophycin C ; II. Optimized Synthesis of Vinyl Sulfonamide Inhibitors of the Cysteine Protease Cruzain
Author: Beth A. Knapp-Reed
Publisher:
ISBN:
Category :
Languages : en
Pages : 474
Book Description
Publisher:
ISBN:
Category :
Languages : en
Pages : 474
Book Description
Modeling, Design and Synthesis of Parasitic Cysteine Protease Inhibitors
Author: Yogesh A. Sabnis
Publisher:
ISBN:
Category :
Languages : en
Pages : 414
Book Description
Publisher:
ISBN:
Category :
Languages : en
Pages : 414
Book Description
Studies Directed Towards the Synthesis of Bafilomycin A1
Author: A. P. Butler
Publisher:
ISBN:
Category :
Languages : en
Pages :
Book Description
Publisher:
ISBN:
Category :
Languages : en
Pages :
Book Description
Total Synthesis of Bafilomycin A1
Author: Florian Karl Kleinbeck
Publisher:
ISBN:
Category :
Languages : en
Pages : 266
Book Description
Publisher:
ISBN:
Category :
Languages : en
Pages : 266
Book Description